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名称：5-氧代-2-氮杂双环[2.2.1]庚烷-2-羧酸叔丁酯

英文名称：TERT-BUTYL 5-OXO-2-AZABICYCLO[2.2.1]HEPTANE-2-CARBOXYLATE

分子式：C11H17NO3

分子量: 211.26
Cas No.：198835-06-2
结构式：

规格：95%

用途：基础原料、有机中间体、医药中间体

合成路线如下：

diborane;

Reactants are commercially availlable.
Slade, David J., US2011/144150, A1, (2011) In a method analogous to J.Malpass and C. Cox, Tetrahedron Lett., 1999, 40, 1419-1422, tert-butyl 2-azabicyclo[2.2.1]hept-5-ene-2-carboxylate is treated with diborane to afford a mixture of alcohols w hich is separated by chromatography.The desired alcohol tert-butyl 5-hydroxy-2-azabicyclo[2.2.1]heptane-2-carboxylate is then oxidized using the Swern procedure to afford the title compound.